Discovery of indole-piperazine derivatives as selective histone deacetylase 6 inhibitors with neurite outgrowth-promoting activities and neuroprotective activities
Ting Liang, Zhao Xie, Baiyun Dang, Jiayun Wang, Tongtong Zhang, Xiaofa Luan, Tao Lu, Chenyu Cao, Xin Chen
Topics & Concepts
ChemistryNeuroprotectionHDAC6Histone deacetylaseNeuriteBenzamideIndole testAcetylationPharmacologyHistone deacetylase inhibitorPiperazineWestern blotBiochemistryIn vitroStereochemistryHistoneBiologyOrganic chemistryGeneHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and AnalysisCholinesterase and Neurodegenerative Diseases