Pyxinol bearing amino acid residues: Easily achievable and promising modulators of P-glycoprotein-mediated multidrug resistance
Conghui Wang, Meng Gao, Shuqi Liu, Zongji Zou, Ruiyin Ren, Chen Zhang, Hao Xie, Jingxian Sun, Yupeng Qi, Qi Qu, Zhihua Song, Gangqiang Yang, Hongbo Wang
Topics & Concepts
ChemistryEffluxP-glycoproteinMultiple drug resistancePaclitaxelTransporterPharmacologyIn vitroAmino acidAmino acid residueStructure–activity relationshipBiochemistryCancerPeptide sequenceBiologyGeneAntibioticsGeneticsDrug Transport and Resistance MechanismsCancer therapeutics and mechanismsGinseng Biological Effects and Applications