Design, synthesis, and biological evaluation of RSL3-based GPX4 degraders with hydrophobic tags
Yao Ning, Zeqi Zhu, Yi‐Cheng Wang, Yi‐Cheng Wang, Xuejing Fan, Jing Wang, Huimei Qian, Xue Qiu, Yong Wang, Yong Wang, Yong Wang
Topics & Concepts
GPX4ChemistryBiochemistryLipid peroxidationGlutathioneEnzymeGlutathione peroxidaseFerroptosis and cancer prognosisPeptidase Inhibition and AnalysisDrug Transport and Resistance Mechanisms