Isoquinolinone derivatives as potent CNS multi-receptor D2/5-HT1A/5-HT2A/5-HT6/5-HT7 agents: Synthesis and pharmacological evaluation
Jian Jin, Kun-Xiao Zhang, Fei Dou, Chao Hao, Yifang Zhang, Xudong Cao, Lanchang Gao, Jiaying Xiong, Xin Liu, Bi‐Feng Liu, Guisen Zhang, Yin Chen
Topics & Concepts
ChemistryCatalepsyPharmacologyhERGDopamine receptor D2Behavioural despair testAntipsychoticDopamineReceptorTail suspension testAtypical antipsychoticSerotoninHaloperidolInternal medicinePsychologyBiochemistrySchizophrenia (object-oriented programming)MedicinePsychiatryPotassium channelHippocampusAntidepressantReceptor Mechanisms and SignalingNeurotransmitter Receptor Influence on BehaviorPharmacological Receptor Mechanisms and Effects