Design, synthesis and biological evaluation of novel indole-3-carboxylic acid derivatives with antihypertensive activity
A. V. Danilenko, Alexander N. Volov, Н. А. Волов, Yana B. Platonova, Serguei V. Savilov
Topics & Concepts
LosartanChemistryIndole testAngiotensin II receptor type 1Angiotensin IICarboxylic acidIn vivoPharmacologyChemical synthesisAngiotensin receptorOral administrationIn vitroRenin–angiotensin systemReceptorBlood pressureBiological activityStereochemistryBiochemistryEndocrinologyMedicineBiologyBiotechnologyReceptor Mechanisms and SignalingInflammatory mediators and NSAID effectsRenin-Angiotensin System Studies