Litcius/Paper detail

CARM1 inhibition reduces histone acetyltransferase activity causing synthetic lethality in CREBBP/EP300-mutated lymphomas

Kylee J. Veazey, Donghang Cheng, Kevin Lin, Oscar D. Villarreal, Guozhen Gao, Mabel Pérez‐Oquendo, Hieu T. Van, Sabrina A. Stratton, Michael R. Green, Han Xu, Yue Lu, Mark T. Bedford, Margarida A. Santos

2020Leukemia56 citationsDOIOpen Access PDF

Topics & Concepts

Histone acetyltransferaseBiologySynthetic lethalityCancer researchCREB-binding proteinAcetyltransferaseMutationHistoneMolecular biologyGeneAcetylationGeneticsDNA repairTranscription factorCREBCancer-related gene regulationEpigenetics and DNA MethylationProtein Degradation and Inhibitors