Discovery of a novel piperlongumine analogue as a microtubule polymerization inhibitor with potent anti-angiogenic and anti-metastatic efficacy
Jinling Qin, LI Hong-liang, Xuan Wang, Yixin Zhang, Yongtao Duan, Yongfang Yao, Hua Yang, Moran Sun
Topics & Concepts
ChemistryAngiogenesisIn vivoTubulinCytotoxicityIn vitroAngiogenesis inhibitorMicrotubuleCell cycleCancer cellMicrotubule polymerizationCell cultureCancer researchApoptosisBiochemistryCancerCell biologyBiologyBiotechnologyGeneticsPiperaceae Chemical and Biological StudiesPhytochemical compounds biological activitiesSynthetic Organic Chemistry Methods