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Hybrid molecules combining GABA-A and serotonin 5-HT6 receptors activity designed to tackle neuroinflammation associated with depression

Monika Marcinkowska, Barbara Mordyl, Nikola Fajkis-Zajączkowska, Agata Siwek, Tadeusz Karcz, Alicja Gawalska, Adam Bucki, Paweł Żmudzki, Anna Partyka, Magdalena Jastrzębska‐Więsek, Bartosz Pomierny, Maria Walczak, Magdalena Smolik, Karolina Pytka, Kamil Mika, Magdalena Kotańska, Marcin Kołaczkowski

2022European Journal of Medicinal Chemistry16 citationsDOIOpen Access PDF

Topics & Concepts

NeuroinflammationChemistryReceptorAntidepressantSerotoninPharmacologySerotonergic5-HT receptorNeurotransmissionIn vivoNeuroscienceInternal medicinePsychologyInflammationBiochemistryHippocampusMedicineBiologyBiotechnologyTryptophan and brain disordersStress Responses and CortisolPharmacological Receptor Mechanisms and Effects
Hybrid molecules combining GABA-A and serotonin 5-HT6 receptors activity designed to tackle neuroinflammation associated with depression | Litcius