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Optimization of 1,4-bis(arylsulfonamido)naphthalene-N,N'-diacetic acids as inhibitors of Keap1-Nrf2 protein-protein interaction to suppress neuroinflammation

Dhulfiqar Ali Abed, Sumi Lee, Wen Xia, Ahmed R. Ali, Vaibhav S. Mangipudy, Lauren M. Aleksunes, Longqin Hu

2021Bioorganic & Medicinal Chemistry16 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryNeuroinflammationKEAP1Oxidative stressCytotoxicityReactive oxygen speciesMicrogliaIn vivoLipopolysaccharideWestern blotTumor necrosis factor alphaBiochemistryInflammationIn vitroPharmacologyTranscription factorGeneImmunologyMedicineBiologyBiotechnologyGenomics, phytochemicals, and oxidative stressTryptophan and brain disordersRedox biology and oxidative stress
Optimization of 1,4-bis(arylsulfonamido)naphthalene-N,N'-diacetic acids as inhibitors of Keap1-Nrf2 protein-protein interaction to suppress neuroinflammation | Litcius