Cross-reactivity to glutamate carboxypeptidase III causes undesired salivary gland and kidney uptake of PSMA-targeted small-molecule radionuclide therapeutics
Laura Lucaroni, Tony Georgiev, Eleonora Prodi, Sara Puglioli, Christian Pellegrino, Nicholas Favalli, Luca Prati, Markus G. Manz, Samuele Cazzamalli, Dario Neri, Sebastian Oehler, Gabriele Bassi
Topics & Concepts
Glutamate carboxypeptidase IIKidneyChemistryImmunofluorescenceRadioligandProstate cancerCancer researchMolecular biologyReceptorBiochemistryAntibodyMedicineInternal medicineBiologyCancerImmunologyProstate Cancer Treatment and ResearchRadiopharmaceutical Chemistry and ApplicationsNeuropeptides and Animal Physiology