The discovery of potent USP2/USP8 dual-target inhibitors for the treatment of breast cancer via structure guided optimization of ML364
Yucheng Tian, Kang Liu, Dongdong Wu, Liuyi Wu, Qianqian Xu, Wei Wei, Zhiyu Li, Qianming Du, Jinlei Bian
Topics & Concepts
ChemistryBreast cancerCancer researchIn vivoCancerPharmacologyInternal medicineMedicineBiologyBiotechnologyUbiquitin and proteasome pathwaysCancer-related Molecular PathwaysPeptidase Inhibition and Analysis