Litcius/Paper detail

Alkylated monoterpene indole alkaloid derivatives as potent P-glycoprotein inhibitors in resistant cancer cells

David Cardoso, Annamária Kincses, Márta Nové, Gabriella Spengler, Silva Mulhovo, João Aires‐de‐Sousa, Daniel J. V. A. dos Santos, Maria‐José U. Ferreira

2020European Journal of Medicinal Chemistry30 citationsDOI

Topics & Concepts

ChemistryIndole testP-glycoproteinStereochemistryLipophilicityMultiple drug resistanceCytotoxicityMonoterpeneDoxorubicinAlkaloidIn vitroBiochemistryPharmacologyChemotherapyBiologyGeneticsAntibioticsDrug Transport and Resistance MechanismsAlkaloids: synthesis and pharmacologyBerberine and alkaloids research