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General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation

Francesca Bartoccini, Fabiola Fanini, Michele Retini, Giovanni Piersanti

2020Tetrahedron Letters10 citationsDOI

Topics & Concepts

Enantiopure drugRegioselectivityChemistryIndole testAlkylationNucleophileTryptophanCombinatorial chemistryMedicinal chemistryStereochemistryOrganic chemistryCatalysisEnantioselective synthesisAmino acidBiochemistryFluorine in Organic ChemistryCatalytic C–H Functionalization MethodsSynthesis and Biological Evaluation
General synthesis of unnatural 4-, 5-, 6-, and 7-bromo-d-tryptophans by means of a regioselective indole alkylation | Litcius