Hydrophobic and polar interactions of FDA-approved small molecule protein kinase inhibitors with their target enzymes
Robert Roskoski
Topics & Concepts
Allosteric regulationSmall moleculeChemistryBiochemistryKinaseDrug discoveryProtein kinase AEnzymeBinding siteProtein Kinase Regulation and GTPase SignalingMelanoma and MAPK PathwaysQuinazolinone synthesis and applications