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Target-based drug discovery, ADMET profiling and bioactivity studies of antibiotics as potential inhibitors of SARS-CoV-2 main protease (Mpro)

Misbaudeen Abdul-Hammed, Ibrahim Olaide Adedotun, Victoria Adeola Falade, Adewusi John Adepoju, Sabitu Babatunde Olasupo, Modinat Wuraola Akinboade

2021VirusDisease75 citationsDOIOpen Access PDF

Topics & Concepts

DrugPharmacologyAntibioticsPharmacokineticsAzithromycinCiprofloxacinBioavailabilityAntiviral drugVirtual screeningDrug discoveryProteaseMedicineComputational biologyChemistryBiologyBioinformaticsMicrobiologyBiochemistryEnzymeComputational Drug Discovery MethodsSARS-CoV-2 and COVID-19 Researchthermodynamics and calorimetric analyses
Target-based drug discovery, ADMET profiling and bioactivity studies of antibiotics as potential inhibitors of SARS-CoV-2 main protease (Mpro) | Litcius