MEN1 mutations mediate clinical resistance to menin inhibition
Florian Perner, Eytan M. Stein, Daniela V. Wenge, Sukrit Singh, Jeonghyeon Kim, Athina Apazidis, Homa Rahnamoun, Disha Anand, Christian Marinaccio, Charlie Hatton, Yanhe Wen, Richard M. Stone, David Schaller, Shoron Mowla, Wenbin Xiao, Holly A. Gamlen, Aaron J. Stonestrom, Sonali Persaud, Elizabeth T. Ener, Jevon Cutler, John G. Doench, Gerard M. McGeehan, Andrea Volkamer, John D. Chodera, Radosław P. Nowak, Eric S. Fischer, Ross L. Levine, Scott A. Armstrong, Sheng F. Cai
Topics & Concepts
ChromatinBiologyCancer researchMutationBRD4Gene mutationSomatic cellMEN1Chromatin remodelingGeneticsGeneBromodomainEpigeneticsMultiple endocrine neoplasiaProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsChronic Lymphocytic Leukemia Research