Design, synthesis and biological evaluation of rasagiline-clorgyline hybrids as novel dual inhibitors of monoamine oxidase-B and amyloid-β aggregation against Alzheimer’s disease
Sai‐Sai Xie, Jing Liu, Chunli Tang, Chengyun Pang, Qing Li, Yuelian Qin, Xiaojie Nong, Zhipeng Zhang, Jie Guo, Maojun Cheng, Weizhong Tang, Ningsheng Liang, Neng Jiang
Topics & Concepts
RasagilineChemistryClorgylineMonoamine oxidase BMonoamine oxidaseIC50PharmacologyMonoamine neurotransmitterPharmacokineticsNeuroprotectionIn vitroBiochemistryEnzymeParkinson's diseaseReceptorDiseaseSerotoninMedicinePathologyAlzheimer's disease research and treatmentsCholinesterase and Neurodegenerative DiseasesMedicinal Plants and Neuroprotection