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Role of Human Arylacetamide Deacetylase (AADAC) on Hydrolysis of Eslicarbazepine Acetate and Effects of AADAC Genetic Polymorphisms on Hydrolase Activity

Keiya Hirosawa, Tatsuki Fukami, Kiyomichi Tashiro, Yoshiyuki Sakai, Fumiya Kisui, Masataka Nakano, Miki Nakajima

2021Drug Metabolism and Disposition23 citationsDOIOpen Access PDF

Topics & Concepts

PhenacetinHydrolysisCarboxylesteraseChemistryPharmacologyProdrugMicrosomeBiochemistryEnzymeBiologyPharmacological Effects and Toxicity StudiesCholinesterase and Neurodegenerative DiseasesBipolar Disorder and Treatment
Role of Human Arylacetamide Deacetylase (AADAC) on Hydrolysis of Eslicarbazepine Acetate and Effects of AADAC Genetic Polymorphisms on Hydrolase Activity | Litcius