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Predicting budesonide performance in healthy subjects and patients with Crohn's disease using biorelevant in vitro dissolution testing and PBPK modeling

Angela Effinger, Caitríona M. O’Driscoll, Mark McAllister, Nikoletta Fotaki

2020European Journal of Pharmaceutical Sciences28 citationsDOI

Topics & Concepts

Physiologically based pharmacokinetic modellingBudesonideBioavailabilityPharmacokineticsPharmacologyDrugPopulationChemistryCYP3A4MedicineInternal medicineCorticosteroidCytochrome P450MetabolismEnvironmental healthInflammatory Bowel DiseaseHelicobacter pylori-related gastroenterology studiesBiosimilars and Bioanalytical Methods
Predicting budesonide performance in healthy subjects and patients with Crohn's disease using biorelevant in vitro dissolution testing and PBPK modeling | Litcius