Discovery of novel brain-penetrant GluN2B NMDAR antagonists via pharmacophore-merging strategy as anti-stroke therapeutic agents
Qinlong Xu, Mengqi Hu, Jiaming Li, Xiaodong Ma, Zhaoxing Chu, Qihua Zhu, Yanchun Zhang, Panhu Zhu, Yuanzheng Huang, Guangwei He
Topics & Concepts
IfenprodilChemistryNeuroprotectionPharmacologyNMDA receptorMemantineIn vivoAntagonistNeurotoxicityReceptorBiochemistryToxicityMedicineOrganic chemistryBiotechnologyBiologyChemical Synthesis and AnalysisNeuroscience and Neuropharmacology ResearchMolecular Sensors and Ion Detection