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Exploiting the reactivities of<i>ortho</i>-alkynyl aryl ketones: opportunities in designing catalytic annulation reactions

Tian-Shu Zhang, Shuai Liu, Wen‐Juan Hao, Bo Jiang

2022Organic Chemistry Frontiers35 citationsDOI

Abstract

We provide a comprehensive overview of recent progress in this rapidly growing field by summarizing catalytic annulation reactions of ortho -alkynyl aryl ketones which involve carbo- and oxo -cyclization patterns with consideration of their mechanisms and applications.

Topics & Concepts

AnnulationChemistryArylCatalysisCombinatorial chemistryOrganic chemistryMedicinal chemistryAlkylCatalytic C–H Functionalization MethodsCatalytic Alkyne ReactionsCatalytic Cross-Coupling Reactions
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