Litcius/Paper detail

A designed cyclic peptide based on Trastuzumab used to construct peptide-drug conjugates for its HER2-targeting ability

Jiaqi Zhou, Yuxing Zou, Yan Cai, Fanglian Chi, Wenlong Huang, Wei Shi, Hai Qian

2021Bioorganic Chemistry25 citationsDOI

Topics & Concepts

ConjugateCamptothecinTrastuzumabChemistryPeptideMonoclonal antibodyAntibody-drug conjugateOligopeptidePharmacologyAntibodyIn silicoCancer researchBiochemistryCancerBiologyImmunologyMedicineInternal medicineBreast cancerMathematicsGeneMathematical analysisMonoclonal and Polyclonal Antibodies ResearchHER2/EGFR in Cancer ResearchPeptidase Inhibition and Analysis