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Drug antagonism and single-agent dominance result from differences in death kinetics

Ryan Richards, Hannah Schwartz, Megan E. Honeywell, Mariah Stewart, Peter Cruz‐Gordillo, Anna J. Joyce, Benjamin Landry, Michael J. Lee

2020Nature Chemical Biology45 citationsDOIOpen Access PDF

Topics & Concepts

AntagonismDrugDominance (genetics)Programmed cell deathCrosstalkBiologyApoptosisPharmacologyGeneticsReceptorGeneOpticsPhysicsPARP inhibition in cancer therapyComputational Drug Discovery MethodsProtein Structure and Dynamics
Drug antagonism and single-agent dominance result from differences in death kinetics | Litcius