The synthesis, biological evaluation and in silico studies of asymmetric 3,5-diaryl-rhodanines as novel inhibitors of human carbonic anhydrase isoenzymes
Kemal Yararli, Ebru Bilen Ozer, Sinan Bayındır, Cüneyt Çağlayan, Cüneyt Türkeş, Şükrü Beydemir
Topics & Concepts
ChemistryCarbonic anhydraseCarbonic anhydrase IIRhodanineCombinatorial chemistryCatalysisIn silicoStereochemistryEnzymeDocking (animal)Organic chemistryBiochemistryNursingMedicineGeneEnzyme function and inhibitionSynthesis and Catalytic ReactionsCholinesterase and Neurodegenerative Diseases