Elucidation of binding dynamics of tyrosine kinase inhibitor tepotinib, to human serum albumin, using spectroscopic and computational approach
Mohd Amir, Saleem Javed
Topics & Concepts
Human serum albuminChemistryCircular dichroismMolecular dynamicsTyrosine-kinase inhibitorDocking (animal)Protein secondary structureBiophysicsBinding constantQuenching (fluorescence)Molecular bindingBinding siteFluorescenceStereochemistryBiochemistryOrganic chemistryComputational chemistryMoleculeCancerMedicineQuantum mechanicsNursingInternal medicinePhysicsBiologyProtein Interaction Studies and Fluorescence AnalysisLanthanide and Transition Metal ComplexesDrug Transport and Resistance Mechanisms