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Resistance looms for KRAS G12C inhibitors and rational tackling strategies

Junmin Zhang, Juanhong Zhang, Qing Liu, Xing‐Xing Fan, Elaine Lai‐Han Leung, Xiaojun Yao, Liang Liu

2021Pharmacology & Therapeutics54 citationsDOI

Topics & Concepts

KRASClinical trialDrug resistanceMedicineDrug developmentComputational biologyDrugCancerBioinformaticsBiologyPharmacologyInternal medicineGeneticsColorectal cancerProtein Kinase Regulation and GTPase SignalingPI3K/AKT/mTOR signaling in cancerLung Cancer Treatments and Mutations
Resistance looms for KRAS G12C inhibitors and rational tackling strategies | Litcius