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Covalent Binding Mechanism of Furmonertinib and Osimertinib With Human Serum Albumin

Yali Wu, Lili Chen, Jian Chen, Hao Xue, Qingfeng He, Dafang Zhong, Xingxing Diao

2022Drug Metabolism and Disposition20 citationsDOIOpen Access PDF

Topics & Concepts

Human serum albuminChemistryOsimertinibEx vivoPeptideBlood proteinsAlbuminAdductIn vivoBiochemistryIn vitroBiologyReceptorEpidermal growth factor receptorBiotechnologyErlotinibOrganic chemistryChronic Lymphocytic Leukemia ResearchLung Cancer Treatments and MutationsChronic Myeloid Leukemia Treatments
Covalent Binding Mechanism of Furmonertinib and Osimertinib With Human Serum Albumin | Litcius