Development of selective class I protein arginine methyltransferase inhibitors through fragment-based drug design approach
Debomita Bhattacharya, Alice Shi Ming Li, Barnali Paul, Uddipta Ghosh Dastidar, Vijayaratnam Santhakumar, Dipika Sarkar, Irene Chau, Fengling Li, Trisha Ghosh, Masoud Vedadi, Arindam Talukdar
Topics & Concepts
MethyltransferaseChemistryBiochemistryQuinazolineDrug discoveryMethylationArginineDrug developmentSmall moleculeDrug designRational designEnzymeComputational biologyDrugPharmacologyStereochemistryDNABiologyAmino acidGeneticsCancer-related gene regulationEpigenetics and DNA Methylation