Litcius/Paper detail

Development of selective class I protein arginine methyltransferase inhibitors through fragment-based drug design approach

Debomita Bhattacharya, Alice Shi Ming Li, Barnali Paul, Uddipta Ghosh Dastidar, Vijayaratnam Santhakumar, Dipika Sarkar, Irene Chau, Fengling Li, Trisha Ghosh, Masoud Vedadi, Arindam Talukdar

2023European Journal of Medicinal Chemistry13 citationsDOIOpen Access PDF

Topics & Concepts

MethyltransferaseChemistryBiochemistryQuinazolineDrug discoveryMethylationArginineDrug developmentSmall moleculeDrug designRational designEnzymeComputational biologyDrugPharmacologyStereochemistryDNABiologyAmino acidGeneticsCancer-related gene regulationEpigenetics and DNA Methylation