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SC912 inhibits AR-V7 activity in castration-resistant prostate cancer by targeting the androgen receptor N-terminal domain

Qianhui Yi, Xiaojun Han, Henry Yu, Huei-Yu Chen, Dinghong Qiu, Jie Su, Rongtuan Lin, Gerald Batist, Jian Wu

2024Oncogene12 citationsDOI

Topics & Concepts

Androgen receptorProstate cancerCancer researchAntiandrogensAndrogenBiologyAndrogen deprivation therapyApoptosisInternal medicineEndocrinologyCancerMedicineHormoneBiochemistryGeneticsProstate Cancer Treatment and ResearchCancer, Lipids, and MetabolismProtein Degradation and Inhibitors
SC912 inhibits AR-V7 activity in castration-resistant prostate cancer by targeting the androgen receptor N-terminal domain | Litcius