Copper-catalyzed enantioselective arylboronation of activated alkenes leading to chiral 3,3′-disubstituted oxindoles
Jiangfei Chen, Jin‐Heng Li, Yanping Zhu, Qiuan Wang
Abstract
Copper-catalyzed asymmetric arylboronation of activated alkenes for producing highly enantioenriched 3-boroalkyl oxindoles and incorporating pharmacophores is depicted.
Topics & Concepts
ChemistryEnantioselective synthesisCatalysisPharmacophoreCopperCombinatorial chemistryOrganic chemistryStereochemistryCatalytic C–H Functionalization MethodsAxial and Atropisomeric Chirality SynthesisAsymmetric Synthesis and Catalysis