Litcius/Paper detail

Functional Selectivity of a Biased Cannabinoid-1 Receptor (CB<sub>1</sub>R) Antagonist

Ziyi Liu, Malliga R. Iyer, Grzegorz Godlewski, Tony Jourdan, Jie Liu, Nathan J. Coffey, Charles N. Zawatsky, Henry L. Puhl, Jürgen Wess, Jaroslawna Meister, Jeih‐San Liow, Robert B. Innis, Sergio A. Hassan, Yong Sok Lee, George Kunos, Reşat Çınar

2021ACS Pharmacology & Translational Science60 citationsDOIOpen Access PDF

Abstract

R antagonist at reduced risk of central nervous system (CNS) side effects.

Topics & Concepts

RimonabantAntagonistInternal medicineEndocrinologyGene knockdownBiologyAdenylyl cyclasePharmacologyReceptorCell biologyCannabinoid receptorBiochemistryMedicineStimulationGeneCannabis and Cannabinoid ResearchNeuroscience and Neuropharmacology ResearchNeurotransmitter Receptor Influence on Behavior