Litcius/Paper detail

Investigation of the inhibitory activity of some dietary bioactive flavonoids against SARS-CoV-2 using molecular dynamics simulations and MM-PBSA calculations

Jibin K. Varughese, K. L. Joseph Libin, K. S. Sindhu, A. V. Rosily, T. G. Abi

2021Journal of Biomolecular Structure and Dynamics24 citationsDOI

Abstract

is identified as one of the key residue which contributed significantly to MM-PBSA binding energy through hydrophobic interactions. Furthermore, the DFT binding energy values of Amentoflavone (-182.92 kJ/mol) and Naringin (-160.67 kJ/mol) in active site molecular clusters with hydrogen bonds confirmed their potential inhibitory activity. These compounds are of high interest because of their wide availability, low cost, no side effects, and long history of use. We can prevent the severity of this disease for home care patients using these effective dietary supplements. We are hopeful that our results have implications for the development of prophylaxis of COVID-19.Communicated by Ramaswamy H. Sarma.

Topics & Concepts

NaringinChemistryAmentoflavoneMolecular dynamicsProteaseNaringeninInhibitory postsynaptic potentialActive sitePharmacologyStereochemistryBiochemistryComputational chemistryFlavonoidEnzymeMedicineChromatographyAntioxidantInternal medicineBiological Activity of Diterpenoids and BiflavonoidsSynthesis and biological activityComputational Drug Discovery Methods
Investigation of the inhibitory activity of some dietary bioactive flavonoids against SARS-CoV-2 using molecular dynamics simulations and MM-PBSA calculations | Litcius