PARP trapping is governed by the PARP inhibitor dissociation rate constant
Angelica A. Gopal, Bianca Fernandez, Justin Delano, Ralph Weissleder, J. Matthew Dubach
Topics & Concepts
Poly ADP ribose polymerasePARP1PolymeraseDNAChemistryDNA damagePotencyMolecular biologyBiologyBiophysicsCancer researchIn vitroBiochemistryPARP inhibition in cancer therapyDNA Repair MechanismsIntegrated Circuits and Semiconductor Failure Analysis