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PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation

Aleksei E. Machulkin, Anastasia A. Uspenskaya, Nikolay Y. Zyk, Ekaterina A. Nimenko, Anton P. Ber, Stanislav A. Petrov, Radik R. Shafikov, Dmitry A. Skvortsov, Galina B. Smirnova, Yulia A. Borisova, Vadim S. Pokrovsky, Василий Колмогоров, Alexander N. Vaneev, Yan A. Ivanenkov, Alexander D. Khudyakov, С. В. Ковалев, Alexander S. Erofeev, Petr V. Gorelkin, Елена К. Белоглазкина, N. V. Zyk, Elena S. Khazanova, Alexander G. Majouga

2021European Journal of Medicinal Chemistry35 citationsDOIOpen Access PDF

Topics & Concepts

DocetaxelConjugateChemistryPharmacologyPharmacokineticsIn vivoMTT assayCytotoxicityProstate cancerBioavailabilityIn vitroCancerMedicineBiochemistryInternal medicineBiologyMathematicsMathematical analysisBiotechnologyProstate Cancer Treatment and ResearchRadiopharmaceutical Chemistry and ApplicationsMass Spectrometry Techniques and Applications
PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation | Litcius