PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation
Aleksei E. Machulkin, Anastasia A. Uspenskaya, Nikolay Y. Zyk, Ekaterina A. Nimenko, Anton P. Ber, Stanislav A. Petrov, Radik R. Shafikov, Dmitry A. Skvortsov, Galina B. Smirnova, Yulia A. Borisova, Vadim S. Pokrovsky, Василий Колмогоров, Alexander N. Vaneev, Yan A. Ivanenkov, Alexander D. Khudyakov, С. В. Ковалев, Alexander S. Erofeev, Petr V. Gorelkin, Елена К. Белоглазкина, N. V. Zyk, Elena S. Khazanova, Alexander G. Majouga
Topics & Concepts
DocetaxelConjugateChemistryPharmacologyPharmacokineticsIn vivoMTT assayCytotoxicityProstate cancerBioavailabilityIn vitroCancerMedicineBiochemistryInternal medicineBiologyMathematicsMathematical analysisBiotechnologyProstate Cancer Treatment and ResearchRadiopharmaceutical Chemistry and ApplicationsMass Spectrometry Techniques and Applications