Novel coumarin derivatives as multifunctional anti-AD agents: Design, synthesis, X-ray crystal structure and biological evaluation
Ai‐Hong Yang, Hongwei Zhang, Chengting Hu, Xi Wang, Rui Shen, Xiaodi Kou, Huiyan Wang
Topics & Concepts
ChemistryCoumarinAcetylcholinesteraseRational designChelationSelectivityDocking (animal)StereochemistryAntioxidantAchéCombinatorial chemistryIn vitroPopulationIC50EnzymeBiochemistryOrganic chemistryNanotechnologySociologyMedicineNursingCatalysisMaterials scienceDemographyCholinesterase and Neurodegenerative DiseasesAlzheimer's disease research and treatmentsComputational Drug Discovery Methods