Design, synthesis, and pharmacological evaluation of novel 1,2,4-triazol-3-amine derivatives as potential agonists of GABAA subtype receptors with anticonvulsant and hypnotic effects
Reza Jahani, Seyed Reza Abtahi, Manijeh Nematpour, Hossein Fasihi Dastjerdi, Mohsen Chamanara, Zahra Hami, Babak Paknejad
Topics & Concepts
GABAA receptorFlumazenilChemistryPharmacologyAnticonvulsantED50HypnoticZolpidemBenzodiazepineAgonistReceptorAntagonistStereochemistryBiochemistryEpilepsyMedicineNeurosciencePsychologyInsomniaNeuroscience and Neuropharmacology ResearchPhenothiazines and Benzothiazines Synthesis and ActivitiesPharmacological Receptor Mechanisms and Effects