Discovery of a highly selective BChE inhibitor with concomitant anti-neuroinflammatory activity for treating Alzheimer's disease
Yarong Zhao, Kun Wu, Wei Luo, Yuting Zhao, Jing Zeng, Junbo Wu, Changlei Yang, Meiling Yang, Jia‐Bao Liu, Zhengwen Lei, Peng Xue, Zhen Wang
Topics & Concepts
ChemistryPharmacologyConcomitantEnzyme inhibitorButyrylcholinesteraseAlzheimer's diseaseNeuroinflammationDiseaseAchéAcetylcholinesteraseEnzymeBiochemistryInternal medicineMedicineCholinesterase and Neurodegenerative DiseasesTryptophan and brain disordersComputational Drug Discovery Methods