Litcius/Paper detail

Re-evaluating pretomanid analogues for Chagas disease: Hit-to-lead studies reveal both in vitro and in vivo trypanocidal efficacy

Andrew M. Thompson, P. D. T. O’Connor, Andrew J. Marshall, Amanda Fortes Francisco, John M. Kelly, Jennifer Riley, Kevin D. Read, Catherine Perez, Scott Cornwall, Richard C. Thompson, Martine Keenan, Karen L. White, Susan A. Charman, Bilal Zulfiqar, Melissa L. Sykes, Vicky M. Avery, Eric Chatelain, William A. Denny

2020European Journal of Medicinal Chemistry22 citationsDOIOpen Access PDF

Topics & Concepts

Chagas diseaseParasitemiaIn vivoBenznidazoleTrypanosoma cruziTrypanosoma bruceiPharmacologyTrypanocidal agentChemistryIn vitroDrugDosingDrug developmentMalariaBiologyImmunologyParasite hostingBiochemistryPlasmodium falciparumBiotechnologyWorld Wide WebGeneComputer scienceTrypanosoma species research and implicationsResearch on Leishmaniasis StudiesSynthesis and Biological Evaluation