A strategy to discover selective α-glucosidase/acetylcholinesterase inhibitors from five function-similar citrus herbs through LC-Q-TOF-MS, bioassay and virtual screening
Hua Guo, Yuehua Chen, Tian‐Min Wang, Ting‐Guo Kang, Hui-Yang Sun, Wenhan Pei, Hui‐Peng Song, Hui Zhang
Topics & Concepts
ChemistryPharmacophoreAcetylcholinesteraseFlavanoneVirtual screeningTraditional medicineBioassayDocking (animal)Liquid chromatography–mass spectrometryChromatographyEnzymeStereochemistryBiochemistryMass spectrometryFlavonoidAntioxidantBiologyNursingMedicineGeneticsCholinesterase and Neurodegenerative DiseasesPhytochemicals and Antioxidant ActivitiesMedicinal Plants and Neuroprotection