Pharmacokinetic Models Scaled Up from Humanized Liver Mouse Data Can Account for Drug Monitoring Results of Atomoxetine and Its 4-Hydroxylated and N-Demethylated Metabolites in Pediatric Patients Genotyped for Cytochrome P450 2D6
Makiko Shimizu, Shotaro Uehara, Katsuhiro Ohyama, Haruka Nishimura, Yoïchi Tanaka, Yoshiro Saito, Hiroshi Suemizu, Sayaka Yoshida, Hiroshi Yamazaki
Topics & Concepts
AtomoxetineCYP2D6Physiologically based pharmacokinetic modellingPharmacokineticsPharmacologyParoxetineCytochrome P450Atomoxetine hydrochlorideAdverse effectMetaboliteDrugTherapeutic drug monitoringMedicineAttention deficit hyperactivity disorderInternal medicineMethylphenidateMetabolismPsychiatrySerotoninReceptorPharmacogenetics and Drug MetabolismPharmacological Effects and Toxicity StudiesTreatment of Major Depression