Discovery of quinazoline derivatives as a novel class of potent and in vivo efficacious LSD1 inhibitors by drug repurposing
Zhonghua Li, Tingting Qin, Zhongrui Li, Xuan Zhao, Xinhui Zhang, Taoqian Zhao, Nian Yang, Jinxin Miao, Jinlian Ma, Zhenqiang Zhang, Jinlian Ma, Zhenqiang Zhang
Topics & Concepts
ErlotinibChemistryIn vivoPharmacologyDrug repositioningCurcuminIC50ApoptosisCancer researchDrugIn vitroBiochemistryEpidermal growth factor receptorReceptorMedicineBiologyBiotechnologyEpigenetics and DNA MethylationHistone Deacetylase Inhibitors ResearchCancer-related gene regulation