Design, synthesis and mechanistic study of novel diarylpyrazole derivatives as anti-inflammatory agents with reduced cardiovascular side effects
Noha H. Amin, Mohammed I.A. Hamed, Maha M. Abdel‐Fattah, Ahmed H. A. Abusabaa, Mohammed T. El‐Saadi
Topics & Concepts
ChemistryIn vivoPharmacologyADMELactate dehydrogenaseCelecoxibEnzymeIn silicoAnti-inflammatoryDocking (animal)In vitroBiochemistryNursingBiologyBiotechnologyMedicineGeneEicosanoids and Hypertension PharmacologyInflammatory mediators and NSAID effectsOrganic Chemistry Cycloaddition Reactions