Litcius/Paper detail

Design and synthesis of new indole drug candidates to treat Alzheimer’s disease and targeting neuro-inflammation using a multi-target-directed ligand (MTDL) strategy

Phoebe F. Lamie, Maha M. Abdel‐Fattah, John N. Philoppes

2022Journal of Enzyme Inhibition and Medicinal Chemistry28 citationsDOIOpen Access PDF

Abstract

BuChE active sites, drug-likeness, and ADMET prediction were performed.

Topics & Concepts

AchéChemistryIndole testAcetylcholinesteraseIn vitroDrugPharmacologyDocking (animal)SelectivityBiochemistryEnzymeMedicineCatalysisNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments