Synthesis, preclinical evaluation, and a pilot clinical imaging study of [18F]AlF-NOTA-JR11 for neuroendocrine neoplasms compared with [68Ga]Ga-DOTA-TATE
Qing Xie, Teli Liu, Jing Ding, Nina Zhou, Xiangxi Meng, Hua Zhu, Nan Li, Jiangyuan Yu, Zhi Yang
Topics & Concepts
BiodistributionDOTASomatostatin receptor 2ChemistryPet imagingNuclear medicineSomatostatin receptorHigh-performance liquid chromatographyInternalizationSomatostatinMedicineReceptorPositron emission tomographyChromatographyEndocrinologyChelationIn vitroBiochemistryOrganic chemistryNeuroendocrine Tumor Research AdvancesLung Cancer Research StudiesRadiopharmaceutical Chemistry and Applications