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Novel deuterated Mnk1/2 protein degrader VNLG-152R analogs: Synthesis, In vitro Anti-TNBC activities and pharmacokinetics in mice

Puranik Purushottamachar, Elizabeth Thomas, Retheesh S. Thankan, Vincent C.O. Njar

2022European Journal of Medicinal Chemistry12 citationsDOI

Topics & Concepts

ChemistryPharmacokineticsPharmacologyIn vitroPaclitaxelCyclin D1Cancer researchBiochemistryCellCell cycleInternal medicineChemotherapyBiologyMedicineChemical Reactions and IsotopesPharmacogenetics and Drug MetabolismAmino Acid Enzymes and Metabolism
Novel deuterated Mnk1/2 protein degrader VNLG-152R analogs: Synthesis, In vitro Anti-TNBC activities and pharmacokinetics in mice | Litcius