Physiologically based pharmacokinetic combined JAK2 occupancy modelling to simulate PK and PD of baricitinib with kidney transporter inhibitors and in patients with hepatic/renal impairment
Zhongjian Wang, Wei Liu, Xueyan Li, Hong-Jiao Chen, Dongying Qi, Fulu Pan, Huining Liu, Shuang Yu, Bowen Yi, Guopeng Wang, Yang Liu
Topics & Concepts
Physiologically based pharmacokinetic modellingProbenecidPharmacokineticsPharmacologyTransporterPharmacodynamicsKidneyChemistryMedicineUrologyInternal medicineBiochemistryGeneMyeloproliferative Neoplasms: Diagnosis and TreatmentChronic Myeloid Leukemia TreatmentsDrug Transport and Resistance Mechanisms