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Discovery of indol-6-yl-pyrrolo[2,3-c]pyridin-7-one derivatives as bromodomain-containing protein 4 (BRD4) inhibitors for the treatment of kidney fibrosis

Sibei Tao, Shaohua Tao, Fan Guo, Lidan Zhang, Lifeng Zhao, Ping Fu, Liang Ma

2022European Journal of Medicinal Chemistry17 citationsDOIOpen Access PDF

Topics & Concepts

KidneyChemistryFibrosisBRD4PharmacologyKidney diseaseIC50Internal medicineMedicineBiochemistryIn vitroBromodomainAcetylationGeneProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsChromatin Remodeling and Cancer
Discovery of indol-6-yl-pyrrolo[2,3-c]pyridin-7-one derivatives as bromodomain-containing protein 4 (BRD4) inhibitors for the treatment of kidney fibrosis | Litcius