Translating biased agonists from molecules to medications: Serotonin 5-HT1A receptor functional selectivity for CNS disorders
Adrian Newman‐Tancredi, Ronan Depoortère, Mark S. Kleven, Marcin Kołaczkowski, Luc Zimmer
Topics & Concepts
Functional selectivityNeuroscienceSerotonergicAgonistMarmosetReceptorPartial agonistRaphe nucleiSerotoninPharmacologyIntrinsic activityBiologyMedicineInternal medicinePaleontologyReceptor Mechanisms and SignalingNeurotransmitter Receptor Influence on BehaviorNeuroscience and Neuropharmacology Research