Piperazine squaric acid diamides, a novel class of allosteric P2X7 receptor antagonists
Marius Patberg, Andreas Isaak, Friederike T. Füsser, Natalia V. Ortiz Zacarı́as, Laura Vinnenberg, Janine Schulte, Lucia Michetti, Lucie Grey, Cas van der Horst, Petra Hundehege, Oliver Koch, Laura H. Heitman, Thomas Budde, Anna Junker
Topics & Concepts
ChemistryAllosteric regulationPiperazinePharmacologyADMEMoietyPurinergic receptorReceptorStereochemistryDocking (animal)BiochemistryIn vitroBiologyOrganic chemistryNursingMedicineAdenosine and Purinergic SignalingMast cells and histamineAdolescent and Pediatric Healthcare