Litcius/Paper detail

Discovery of 5-bromo-4-phenoxy-N-phenylpyrimidin-2-amine derivatives as novel ULK1 inhibitors that block autophagy and induce apoptosis in non-small cell lung cancer

Dejuan Sun, Zijian Yang, Yongqi Zhen, Yu‐Shang Yang, Yanmei Chen, Yong Yuan, Lan Zhang, Xiaoxi Zeng, Lixia Chen

2020European Journal of Medicinal Chemistry26 citationsDOIOpen Access PDF

Topics & Concepts

PharmacophoreULK1AutophagyChemistryApoptosisAmine gas treatingKinaseLung cancerCancer researchStereochemistryCombinatorial chemistryBiochemistryProtein kinase ABiologyOncologyMedicineOrganic chemistryAMPKAutophagy in Disease and TherapyUbiquitin and proteasome pathwaysChronic Lymphocytic Leukemia Research