Discovery of 5-bromo-4-phenoxy-N-phenylpyrimidin-2-amine derivatives as novel ULK1 inhibitors that block autophagy and induce apoptosis in non-small cell lung cancer
Dejuan Sun, Zijian Yang, Yongqi Zhen, Yu‐Shang Yang, Yanmei Chen, Yong Yuan, Lan Zhang, Xiaoxi Zeng, Lixia Chen
Topics & Concepts
PharmacophoreULK1AutophagyChemistryApoptosisAmine gas treatingKinaseLung cancerCancer researchStereochemistryCombinatorial chemistryBiochemistryProtein kinase ABiologyOncologyMedicineOrganic chemistryAMPKAutophagy in Disease and TherapyUbiquitin and proteasome pathwaysChronic Lymphocytic Leukemia Research